Dr. Y. V. D. Nageswar, FRSC Coordinator for PhD Programme NIPER-Hyderabad

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1 Dr. Y. V. D. Nageswar, FRSC Coordinator for PhD Programme NIPER-Hyderabad QUALIFICATION - M.Sc., Ph.D., (Organic Chemistry), P.G.D.P.M, P.G.D.HRM., P.G.DEM EXPERIENCE - 33 years of research experience in synthetic organic chemistry AREA OF RESEARCH INTEREST - Medicinal Chemistry - Green Chemistry - Supramolecular Chemistry - Nano catalysis AWARDS AND HONORS - Fellow of Royal Society of Chemistry, London (FRSC) - Fellow of Association of Biotechnology and Pharmacy (FABP) - Fellow of Indian Council of Chemists (FICC). - Fellow of Indian Chemical Society (FICS), Kolkata - Merit certificate received for successful commercialization of mefloquine process for the first time - Best performance award , , from IICT CURRENT MEMBERSHIP OF PROFESSIONAL BODIES - Life member Indian Society for Analytical Scientists (ISAS) - Life Member, Oil Technologists Association of India (OTAI) - Life Member, Indian Pharmacological Society (IPS) - Life Member, Indian Institute of Chemical Engineers (IIChE) LIST OF PUBLICATIONS (Last Five Years) 1. Novel and efficient supramolecular synthesis of pyrroles in the presence of β-cyclodextrin in water. K. Ramesh, K. Karnakar, G. Satish, Y.V.D. Nageswar. Chinese Chemical Letters, 23, 1331, A concise aqueous phase supramolecular synthesis of 2-phenyl-2,3-dihydroquinazolin-4(1H)-one derivatives, K. Ramesh, K. Karnakar, G. Satish, B.S.P. Anil Kumar, Y.V.D. Nageswar. Tetrahedron Letters, 53, 6936, Recyclable Ru/C catalyzed oxidative cyanation of tertiary amines with TBHP. K. Harsha Vardhan Reddy, G. Satish, V. Prakash Reddy, B. S. P. Anil Kumar, Y. V. D. Nageswar. RSC Advances, 2, 11084, Tandem supramolecular synthesis of substituted 2-aryl-2, 3-dihydroquinazolin-4(1H)-ones in the presence of β-cyclodextrin in water. K. Ramesh, K. Karnakar, G. Satish, K. Harsha Vardhan Reddy, Y. V. D. Nageswar. Tetrahedron Letters, 53, 6095, A simple, solvent and catalyst-free green synthetic protocol for β-amino phosphonates. K. Ramesh, S. Narayana Murthy, K. Karnakar, Y. V. D. Nageswar. Eur. J. Chem, 3, 119,

2 6. Recyclable graphite oxide promoted efficient synthesis of 2-phenyl quinozoline derivatives in the presence of TBHP as an oxidant. K. Karnakar, A. Vijay Kumar, S. Narayana Murthy, K. Ramesh, Y. V. D. Nageswar. Tetrahedron Letters, 53, 4613, Magnetically separable CuFe 2 O 4 nano particles catalyzed multicomponent synthesis of 1,4-disubstituted 1,2,3-triazoles in tap water using click chemistry B. S. P. Anil Kumar, K. Harsha Vardhan Reddy, B. Madhav, K. Ramesh, Y. V. D. Nageswar. Tetrahedron Letters, 53, 4595, A tandem one pot aqueous phase synthesis of thiazoles/selenazoles, B. Madhav, S. Narayana Murthy, B. S. P. Anil Kumar, K. Ramesh, Y. V. D. Nageswar. Tetrahedron Letters, 53, 3835, Magnetically separable CuFe 2 O 4 Nanoparticles catalysed C-Se cross-coupling in Reusable PEG medium. K. Harsha Vardhan Reddy, G. Satish, K.Ramesh, K. Karnakar. Y. V. D. Nageswar. Chemistry Lett. 41, 585, Simple and straight forward synthesis of 2,4-disubstituted quinazolines in aqueous medium. B. Madhav, S. N. Murthy, B. S.P A. Kumar, A. A. Kumar and Y. V. D. Nageswar Eur. J. Chem, 3, 252, A novel one-pot synthesis of spiro[indoline-3,4 -pyrazolo[3,4-e][1,4]thiazepine] diones using recyclable bioglycerol-based sulfonic acid functionalized carbon catalyst. K. Karnakar, S. Narayana Murthy, K. Ramesh, K. Harsha Vardhan Reddy Y.V.D. Nageswar U. Chandrakala, B.L.A. Prabhavathi Devi, R.B.N. Prasad. Tetrahedron Letters, 53, 3497, An efficient synthesis of N-substituted indoles from indoline/indoline carboxylic acid via aromatization followed by C N cross-coupling reaction by using nano copper oxide as a recyclable catalyst. K. Harsha Vardhan Reddy, G. Satish, K. Ramesh, K. Karnakar, Y.V.D. Nageswar. Tetrahedron Letters, 53, 3061, Polyethylene glycol (PEG-400): an efficient and recyclable reaction medium for the synthesis of pyrazolo[3,4-b]quinoline derivatives. K. Karnakar, S. Narayana Murthy, K. Ramesh, G. Satish, Jagadeesh Babu Nanubolu, Y.V.D. Nageswar, Tetrahedron Letters, 53, 2897, Synthesis of N- substituted pyrroles under catalyst and solvent free conditions. K. Ramesh, S. N. Murthy, Y. V. D. Nageswar. Synth. Commun., 42, 2471, A mild and expeditious synthesis of amides from aldehydes using bio glycerol-based carbon as a recyclable catalyst. K. Ramesh, S. Narayana Murthy, K. Karnakar, K. Harsha Vardhan Reddy, Y.V.D. Nageswar, M. Vijay, B.L.A. Prabhavathi Devi, R.B.N. Prasad. Tetrahedron Letters, 53, 2636, Synthesis of 2-N-substituted benzothiazoles via domino condensation-hetero cyclization process, mediated by copper oxide nanoparticles under ligand-free conditions G. Satish, K. Harsha Vardhan Reddy, K. Ramesh, K. Karnakar, Y.V.D. Nageswar, Tetrahedron Letters, 53, 2518, A novel bioglycerol-based recyclable carbon catalyst for an efficient one-pot synthesis of highly substituted imidazoles. K. Ramesh, S. Narayana Murthy, K. Karnakar, Y.V. D. Nageswar,, Kukuma Vijayalakhshmi, Bethala L.A. Prabhavathi Devi, R.B.N. Prasad Tetrahedron Letters, 53, 1126, A facile, aqueous phase green synthetic protocol for the synthesis of 5,9b-dihydro-1H-[1,2,4]triazino[5, 6-b]indole-3-ols/5,9b-dihydro-1H-[1,2,4]triazino[5, 6-b]indole-3-thiols.K. Ramesh, S. Narayana Murthy, K. Karnakar, Y.V. D. Nageswar, Tetrahedron Letters, 52,,4734, o-iodoxybenzoic acid(ibx):a versatile reagent for the synthesis of N-substituted pyrroles mediated by β-cyclodextrin in water. S. Narayana Murthy, Y.V.D. Nageswar. Tetrahedron Letters, 52,,4481, DABCO-promoted three-component reaction between amines, dialkyl acetylenedicarboxylates, and glyoxal. K. Ramesh, S. Narayana Murthy, K. Karnakar, Y. V. D. Nageswar Tetrahedron Letters, 52, 3937,

3 21. Recyclable Heterogeneous Copper Oxide On Alumina Catalyzed Coupling of Phenols and Alcohols with Aryl halides under Ligand Free Conditions. K. Swapna, S. N. Murthy, M.T. Jyothi, Y. V. D. Nageswar. Org. Bio. Chem. 9, 5978, Nano CuFe 2 O 4 as a Magnetically Separable and Reusable Catalyst for the Synthesis of Diaryl/Aryl Alkyl sulfides via Cross-Coupling process under Ligand Free Conditions. K. Swapna, S. N. Murthy, M.T. Jyothi, Y. V. D. Nageswar. Org. Bio. Chem. 9, 5989, Optimization of nitrilase production from Alcaligenes faecalis MTCC (IICT-A3): effect of inducers on substrate specificity. Y. V. D. Nageswar, Gurrala Sheelu, Rekha Rao Shambhu, Hemalatha Muluka, Nooreen Mehdi, M. Shaheer Malik, Ahmed Kamal. Bioprocess Biosyst Eng 34, 515, Nano copper oxide catalyzed synthesis of symmetrical diaryl sulfides under ligand free conditions. K, Harsha vardhan Reddy, V. Prakash Reddy, A. Ashwan Kumar, G. Kranthi. Y. V. D. Nageswar, Beilstein J. Org. Chem. 7, 886, Nano Copper Oxide Catalyzed Synthesis of Symmetrical Diaryl Selenides Via Cascade Reaction of KSeCN with Aryl Halides K, Harsha vardhan Reddy, V.Prakash Reddy, B, Madhav, J. Shankar. Y. V. D. Nageswar. Synlett., 9, 1268, An Efficient Protocol for the Synthesis of 2-Phenylquinazolines Catalyzed by Ceric Ammonium Nitrate (CAN). K. Karnakar, J.Shankar, S. Narayana Murthy, K, Ramesh, Y. V. D. Nageswar. Synlett., 8, 1089, Quinoxaline synthesis in novel tandem one-pot protocol. B.S.P.Anil Kumar, B, Madhav, K, Harsha vardhan Reddy, Y. V. D. Nageswar. Tetrahedron Lett., 52, 2862, Copper oxide nanoparticles catalyzed synthesis of aryl sulfides via cascade reaction of aryl halides. K, Harsha vardhan Reddy, V.Prakash Reddy, J.Shankar, B, Madhav, B.S.P.Anil Kumar, Y. V. D. Nageswar. Tetrahedron Lett., 52, 32679, Novel and efficient aqueous phase synthesis of N-substituted azephines via tandem Michael addition and cyclization in the presence of β-cyclodextrin. K, Ramesh, S. Narayana Murthy, Y. V. D. Nageswar. Tetrahedron Lett., 52, 2362, Magnetically Separable and Reusable Copper Ferrite Nano Particles for Cross Coupling of Aryl Halides with Diphenyl Diselenide. K. Swapna, S. N. Murthy, Y. V. D. Nageswar. Eur. J. Org. Chem. 1940, Synthesis of Allyl aryl sulfones from the Baylis-Hillman acetates in water. K. Karnakar, J. Shankar, S. N. Murthy, Y. V. D. Nageswar. Helv. Chim. Acta., 2011, 94, Aqueous phase synthesis of α-hydroxy phosphonates catalyzed by β-cyclodextrin. K. Ramesh, B. Madhav, S. N. Murthy, Y. V. D. Nageswar. Synth. Commun., 42, 258, Stereoselective Formal Total Synthesis of ( )-Swainsonine from Garner s Aldehyde. S. N. Murthy, Y. V. D. Nageswar. Synthesis 755, A New, Efficient and Recyclable Lanthanum (III) Oxide Catalyzed C-N Cross-Coupling. S. N. Murthy, B. Madhav, V. P. Reddy, Y. V. D. Nageswar. Adv. Synth. Catal. 352, 3241, Copper Iodide as a Recyclable Catalyst for Buchwald N-arylation. K. Swapna, S. N. Murthy, Y. V. D. Nageswar. Eur. J. Org. Chem., 6678, MnCl 2 4H 2 O Catalyzed Potential Protocol for the Synthesis of Aryl/vinyl Sulfides. B. Madhav, S. N. Murthy, K. Ramesh, Y. V. D. Nageswar. Chem. Lett., 39, 1149,

4 37. One-pot synthesis of 2-amino-4H-chromen-4-yl phosphonate derivatives using β-cyclodextrin as reusable catalyst in water. S. N. Murthy, B. Madhav, V. Prakash Reddy, Y. V. D. Nageswar. Tetrahedron Lett., 51, 3649, DABCO as a mild and efficient catalytic system for the synthesis of highly substituted imidazoles via multi-component condensation strategy. S. N. Murthy, B. Madhav, Y. V. D. Nageswar. Tetrahedron Lett., 51, 5252, An Improved Protocol for the Synthesis of Quinoline-2, 3-dicarboxylates Under Neutral Conditions via Biomimetic Approach. B. Madhav, S. N. Murthy, K. R. Rao, Y. V. D. Nageswar. Helv. Chim. Acta. 93, 257, Revisiting the Hinsberg Reaction: Facile and Expeditious Synthesis of 3-Substituted Quinoxalin-2(1H)- ones under Catalyst-Free Conditions in Water. S. N. Murthy B. Madhav, Y. V. D. Nageswar. Helv. Chim. Acta. 93, 1216, Novel aqueous phase supramolecular synthesis of α -oxindole-α-hydroxyphosphonates. J.Shankar, K.Karnakar, B.Srinivas, Y. V. D. Nageswar. Tetrahedron Lett., 51, 3938, Antimicrobial activity from the extracts of fungal isolates of soil and drug samples from Kaziranga national Park, Assam, India C.Ganesh Kumar, P. Mongolla, J. Joseph, Y. V. D. Nageswar. J.mycmed. 20, 283, Multi-Component Supramolecular Synthesis of Spirooxiindoles Catalysed by - cyclodextrin in Water. R. Sridhar, B. Srinivas, B. Madhav, V. P. Reddy, Y. V. D. Nageswar, K. R. Rao. Can. J. Chem. 1704, Lanthanum (III) Oxide as a Recyclable Catalyst for the Synthesis of Diaryl Sulfides and Diaryl Selenides. S. N. Murthy, B. Madhav, V. P. Reddy, Y.V. D. Nageswar. Eur. J. Org. Chem., 5902, Facile and efficient synthesis of 3, 4, 5-substituted furan-2(5h)-ones by using β-cyclodextrin as reusable catalyst. S. N. Murthy, B. Madhav, A. V. Kumar, K. R. Rao, Y. V. D. Nageswar. Tetrahedron, 65, 5251, Biomimetic synthesis of quinoxalines in water. B. Madhav, S. N. Murthy, V. P. Reddy, K. R. Rao, Y. V. D. Nageswar. Tetrahedron Lett., 50, 6025, An approach toward the synthesis of β-hydroxy sulfones on water. S. N. Murthy, B. Madhav, V. P. Reddy, Y. V. D. Nageswar. Tetrahedron Lett., 50, 5009, Multicomponent Approach towards the Synthesis of Substituted Pyrroles under Supramolecular Catalysis Using -Cyclodextrin as a Catalyst in Water under Neutral Conditions. S. N. Murthy, B. Madhav, A.V. Kumar, K. R. Rao, Y. V. D. Nageswar. Helv. Chim. Acta, 92, 2118, Cyclodextrin promoted addition of benzene-selenol to conjugated alkenes in water R. Sridhar, B. Srinivas, Y. V. D. Nageswar, K. R. Rao. Helv. Chim. Acta. 92, 1080, Modified cyclodextrins as enantioselective hosts for amino acids. V. Pavan Kumar, I. Suryanarayana, Y. V. D. Nageswar, K. Rama Rao. Helv. Chim. Acta, 91, 753, Chiral Discrimination of Tolterodine Tartrate by Modified Cyclodextrins. V.PavanKumar, I. Suryanarayana, Y. V. D. Nageswar, K. Rama Rao. J. Carbohydr.Chem., 27, 223, REVIEWS, BOOK CHAPTERS AND BOOKS 1. Supramolecular catalysis of organic reactions involving cyclodextrins (P ) Advances in Organic Synthesis, Vol.1. K.Rama Rao, Y. V. D. Nageswar, N. Srilakshmi Krishnaveni, K. Surendra. Ed. Attaur-Rahman, published by Bentham Science Publishers Ltd.( (Book Chapter- invited) 4

5 2. Cyclodextrins as Promoters in Aqueous Organic Synthesis. K. R. Rao, Y. V. D. Nageswar, R. Sridhar, V. P. Reddy. Current Organic Chemistry, 14, 1308, (Review article-invited) 3. Recent Advances in Biomimetic Synthesis Involving Cyclodextrins.Y. V. D. Nageswar, S. N. Murthy, B. Madhav, J. Shankar. A chapter in Advances in Biomimetics published by INTECH. (Book Chapter- invited) (Ch.5, Page No ). 4. Advances in the Synthesis of Heterocyclic Compounds in Aqueous Medium. Y. V. D. Nageswar, K, Harsha Vardhan Reddy, S. Narayana Murthy, A, Aswan Kumar. A chapter in Water condensation: processes, modelling, control published by NOVA Science publishers, New York (Book Chapterinvited) (Ch.4, Page No ). 5. Recent Research Developments in Foldamer Chemistry published by NOVA Science publishers, New York. Editor Y. V. D. Nageswar. 6. Recent Advances in Materials for Organic Light Emitting Devices published by Research Signpost, India. (in press) PATENTS 1. A process for synthesis of 1-(aryloxy) propionyl-2-arylsulfonyl hydrazines as new hypoglycemic agents. T. Ramalingam, Y. V. D. Nageswar, S. Ramakrishna, A. Bhaskar Rao, P. V. Diwan, J. S. Yadav and K. V. Raghavan. Indian Patent Appl. no. 379/DEL/ A novel synthesis of 1-(aryloxy) propionyl-2-arylsulfonyl hydrazines as new hypoglycemic agents. T. Ramalingam, Y. V. D. Nageswar, S. Ramakrishna, A. Bhaskar Rao, P. V. Diwan, J. S. Yadav and K. V. Raghavan. Indian Patent. Appl. no. 378/DEL/ A process for synthesis of new heterocyclic substituted sulfamides as new anti bacterial agents. K. Rama Rao, Y. V. D. Nageswar, J. S. Yadav, Kaiser Jamil, P. Srinivas Reddy. Indian Patent. Appl. no. 578/DEL/ Process for the preparation of 4-bromo or 4- iodo, 2, 8-bis (trifluoromethyl) quinoline. Y. V. D. Nageswar, H. M. Meshram, P. B. Sattur. Indian Patent. No Improved process for the preparation of the 2-pyridyl, 2, 8-bis (trifluoromethyl)-4-quinoline methanol. Y. V. D. Nageswar, H. M. Meshram, P. B. Sattur. Indian Patent. No Improved process for the preparation of mefloquine hydrochloride. Y. V. D. Nageswar, H. M. Meshram, P. B. Sattur. Indian Patent. No Process for the preparation of 4-cycano- 2, 8-bis(trifluoromethyl) quinoline. Indian Patent. Y. V. D. Nageswar, H. M. Meshram, A. R. Prasad, P. B. Sattur. Indian Patent. No Process for the preparation of the 2-pyridyl, 2, 8-bis (trifluoromethyl)-4-quinolyl ketone. Y. V. D. Nageswar, H. M. Meshram, A. R. Prasad, S. R. Hashim, P. B. Sattur. Indian Patent. No Improved process for the preparation of mefloquine hydrochloride. Y. V. D. Nageswar, H. M. Meshram, A. R. Prasad, S. R. Hashim, P. B. Sattur. Indian Patent. No Improved process for the preparation of mefloquine hydrochloride. Y. V. D. Nageswar, H. M. Meshram, A. R. Prasad, S. R. Hashim, P. B. Sattur. Indian Patent. No Process for the preparation of 4-tosyloxy-, 2, 8-bis (trifluoromethyl) quinoline. Y. V. D. Nageswar, H. M. Meshram, P. B. Sattur. Indian Patent. No

6 12. Improved process for the preparation of the 2-pyridyl, 2, 8-bis (trifluoromethyl)-4-quinolyl ketone. Y. V. D. Nageswar, H. M. Meshram, P. B. Sattur, A. R. Prasad, S. R. Hashim. Indian Patent. No A process for the preparation of alkali and alkaline earth metal salts of substituted ά-(3-pentadecyl phenoxy) isobutyric acid. T. Ramalingam, Y. V. D. Nageswar, M. V. Rao, P. B. Sattur, G. Thyagarajan. Indian Patent. No. 160, Novel hypolipidemic and hypocholesteremic compounds and their preparation and use. T. Ramalingam, Y. V. D. Nageswar, M. V. Rao, P. B. Sattur, G. Thyagarajan. European Patent. No. EP 244, Novel therapeutic compounds useful as hypolipidemic and hypocholesteremic agents and process for the preparation thereof. T. Ramalingam, Y. V. D. Nageswar, M. V. Rao, P. B. Sattur, G. Thyagarajan. US patent. No Novel therapeutic compounds useful as hypolipidemic and hypocholesteremic agents and process for the preparation thereof. T. Ramalingam, Y. V. D. Nageswar, M. V. Rao, P. B. Sattur, G. Thyagarajan. Australian patent. No A process for the preparation of substituted (1-methyl-2-pyrrolidinylidene)-sulfamides. K. Rama Rao, Y. V. D. Nageswar, P. V. Diwan, A. B. Rao, P. B. Sattur, G. Thyagarajan. Indian Patent. No. 635 / A process for the preparation of substituted (1-methyl-2-pyrrolidinylidene)-sulfamides. K. Rama Rao, Y. V. D. Nageswar, P. V. Diwan, A. B. Rao, P. B. Sattur, G. Thyagarajan. Indian Patent. No. 655 / 6